Product Name |
Acenocoumarol-d5 |
Alternate Names |
Acenocoumarol Stable Isotopes, Stable Isotopes of Acenocoumarol |
CAT No. |
CS-BR-00001
|
CAS No. |
152-72-7(Unlabeled) |
Category |
Stable Isotopes |
Stock |
Enquire
|
Mol. Wt. |
Not Available |
Mol. For. |
Not Available
|
Hazardous |
This is not a Hazardous Compound
|
COA |
View Sample COA
|
MSDS |
View Sample MSDS
|
Parent API |
Acenocoumarol |
Smileys |
CC(CC(C(C([2H])=C1[2H])=C(C([2H])=C1[N](=O)=O)[2H])([2H])C(C2=O)=C(C3=CC=CC=C3O2)O)=O |
Controlled |
No |
Shipping |
Free for purchase above 1000$ |
Delivery |
In-Stock, products will be dispatched within 24 hours via FedEx for USA, Europe, and other countries. |
Return |
Returns/replacement accepted if you are not satisfied with the quality of the product, (please send us an email with the reason/issues which are facing, within 15 days, after receipt of the product). |
Ordering |
Place your order online or by email sales@clearsynth.com |
If you find a better price anywhere else we guarantee Price match.
Acenocoumarol-d5 is a deuterated form of acenocoumarol, which is a coumarin derivative used as an oral anticoagulant medication. It is primarily prescribed for the prevention and treatment of thromboembolic disorders, including deep vein thrombosis, pulmonary embolism, and stroke. Acenocoumarol-d5 works by inhibiting the vitamin K-dependent clotting factors in the liver, thus preventing the formation of blood clots.
Chemically, acenocoumarol-d5 is a racemic mixture of two enantiomers, S-(+)-acenocoumarol and R-(-)-acenocoumarol, both of which are deuterated at the 5-position of the coumarin ring. The deuterium labeling is used for pharmacokinetic studies, as it allows for the differentiation of the labeled drug from the endogenous compound and provides more accurate measurements of drug concentrations in biological samples.
Acenocoumarol-d5 is typically administered orally in tablet form and is metabolized in the liver by cytochrome P450 enzymes. The drug has a long half-life of approximately 8-11 hours and requires careful monitoring of blood clotting parameters to ensure therapeutic efficacy and avoid bleeding complications.
Overall, acenocoumarol-d5 is an important medication for the prevention and treatment of thromboembolic disorders, and its deuterium labeling provides valuable insights into its pharmacokinetics and metabolism.